Gary Pitt-Publications

Gary Pitt-Publications

Researcher: 

Selected publications

  1. Stokes NR, Baker N, Bennett JM, Chauhan PK, Collins I, Davies DT, Gavade M, Kumar D, Lancett P, Macdonald R, Macleod L, Mahajan A, Mitchell JP, Nayal N, Nayal YN, Pitt GR, Singh M, Yadav A, Srivastava A, Czaplewski LG, Haydon DJ. Design, synthesis and structure-activity relationships of substituted oxazole-benzamide antibacterial inhibitors of FtsZ. Bioorg Med Chem Lett 2014, 24 (1), 353-9 PMID: 24287381
  2. Palmer JT, Axford LC, Barker S, Bennett JM, Blair M, Collins I, Davies DT, Ford L, Gannon CT, Lancett P, Logan A, Lunniss CJ, Morton CJ, Offermann DA, Pitt GR, Rao BN, Singh AK, Shukla T, Srivastava A, Stokes NR, Thomaides-Brears HB, Yadav A, Haydon DJ. Discovery and in vivo evaluation of alcohol-containing benzothiazoles as potent dual-targeting bacterial DNA supercoiling inhibitors. Bioorg Med Chem Lett 2014, 24 (17), 4215-4222. PMID: 25086682
  3. Axford LC, Agarwal PK, Anderson KH, Andrau LN, Atherall J, Barker S, Bennett JM, Blair M, Collins I, Czaplewski LG, Davies DT, Gannon CT, Kumar D, Lancett P, Logan A, Lunniss CJ, Mitchell DR, Offermann DA, Palmer JT, Palmer N, Pitt GR, Pommier S, Price D, Narasinga Rao B, Saxena R, Shukla T, Singh AK, Singh M, Srivastava A, Steele C, Stokes NR, Thomaides-Brears HB, Tyndall EM, Watson D, Haydon DJ. Design, synthesis and biological evaluation of alpha-substituted isonipecotic acid benzothiazole analogues as potent bacterial type II topoisomerase inhibitors. Bioorg Med Chem Lett 2013, 23 (24), 6598-603. PMID: 24239017
  4. Yea CM, Allan CE, Ashworth DM, Barnett J, Baxter AJ, Broadbridge JD, Franklin RJ, Hampton SL, Hudson P, Horton JA, Jenkins PD, Penson AM, Pitt GR, Rivière P, Robson PA, Rooker DP, Semple G, Sheppard A, Haigh RM, Roe MB. New benzylureas as a novel series of potent, nonpeptidic vasopressin V2 receptor agonists. J Med Chem 2008, 51 (24), 8124-34. PMID: 19053774
  5. Ashworth DM, Batt AR, Baxter AJ, Broqua P, Haigh RM, Hudson P, Heeney CMS, Laporte R, Penson A, Pitt GRW, Robson PA, Rooker DP, Tartar AL, Yea CM, Roe MB. Nonpeptide oxytocin agonists. Drugs Fut 2006, 31 (4), 345-353. Reference
  6. Pitt GR, Batt AR, Haigh RM, Penson AM, Robson PA, Rooker DP, Tartar AL, Trim JE, Yea CM, Roe MB. Non-peptide oxytocin agonists. Bioorg Med Chem Lett 2004, 14 (17), 4585-9. PMID: 15357997
  7. Semple G, Ashworth DM, Batt AR, Baxter AJ, Benzies DW, Elliot LH, Evans DM, Franklin RJ, Hudson P, Jenkins PD, Pitt GR, Rooker DP, Yamamoto S, Isomura Y. Peptidomimetic aminomethylene ketone inhibitors of interleukin-1 beta-converting enzyme (ICE). Bioorg Med Chem Lett 1998, 8 (8), 959-64. PMID: 9871520
  8. Evans DM, Jones DM, Pitt GR, Sueiras-Diaz J, Horton J, Ashworth D, Olsson H, Szelke M. Selective inhibitors of plasma kallikrein. Immunopharmacology 1996, 32 (1-3), 115-6. PMID: 8796284
  9. Evans DM, Jones DM, Pitt GR, Ashworth D, De Clerck F, Verheyen F, Szelke M. Synthetic inhibitors of human tissue kallikrein. Immunopharmacology 1996, 32 (1-3), 117-8. PMID: 8796285